KENPAULLONE
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- $27 - $1802
- Product name: KENPAULLONE
- CAS: 142273-20-9
- MF: C16H11BrN2O
- MW: 327.18
- EINECS:
- MDL Number:MFCD02683595
- Synonyms:9-Bromo-7,12-dihydro-indolo[3,2-d][1]benzazepin-6(5H)-one, NSC 664704;9-BroMopaullone;Kenpaullon;9-BROMO-7,12-DIHYDRO-INDOLO[3,2-D][1]BENZAZEPIN-6(5H)-ONE;8-BROMO-7,12-DIHYDRO-INDOLO[3,2-D][1]-BENZAZEPIN-6(5H)-ONE;KENPAULLONE;NSC-664704;Kenpaullone 9-Bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one
48 prices
Selected condition：
Brand
- AK Scientific
- Ambeed
- ApexBio Technology
- Arctom
- Biorbyt Ltd
- Biosynth Carbosynth
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- Tocris
- TRC
- Usbiological
Package
- 10mM(in 1mL DMSO)
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 10
- 100mg
- 250mg
- 1g
- ManufacturerAK Scientific
- Product numberX5716
- Product descriptionKenpaullone
- Packaging50mg
- Price$197
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging1mg
- Price$27
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging5mg
- Price$46
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging10mg
- Price$60
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging50mg
- Price$102
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging100mg
- Price$164
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging250mg
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA196851
- Product descriptionKenpaullone 98+%
- Packaging1g
- Price$634
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6720
- Product descriptionKenpaullone
- Packaging5mg
- Price$105
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6720
- Product descriptionKenpaullone
- Packaging10mM(in 1mL DMSO)
- Price$116
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6720
- Product descriptionKenpaullone
- Packaging10mg
- Price$162
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberB6720
- Product descriptionKenpaullone
- Packaging50mg
- Price$570
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS025643
- Product descriptionKenpaullone ≥98%
- Packaging1mg
- Price$27
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS025643
- Product descriptionKenpaullone ≥98%
- Packaging5mg
- Price$46
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS025643
- Product descriptionKenpaullone ≥98%
- Packaging10mg
- Price$59
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS025643
- Product descriptionKenpaullone ≥98%
- Packaging50mg
- Price$101
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | X5716 | Kenpaullone | 50mg | $197 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 1mg | $27 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 5mg | $46 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 10mg | $60 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 50mg | $102 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 100mg | $164 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 250mg | $245 | 2021-12-16 | Buy |
| Ambeed | A196851 | Kenpaullone 98+% | 1g | $634 | 2021-12-16 | Buy |
| ApexBio Technology | B6720 | Kenpaullone | 5mg | $105 | 2021-12-16 | Buy |
| ApexBio Technology | B6720 | Kenpaullone | 10mM(in 1mL DMSO) | $116 | 2021-12-16 | Buy |
| ApexBio Technology | B6720 | Kenpaullone | 10mg | $162 | 2021-12-16 | Buy |
| ApexBio Technology | B6720 | Kenpaullone | 50mg | $570 | 2021-12-16 | Buy |
| Arctom | AS025643 | Kenpaullone ≥98% | 1mg | $27 | 2021-12-16 | Buy |
| Arctom | AS025643 | Kenpaullone ≥98% | 5mg | $46 | 2021-12-16 | Buy |
| Arctom | AS025643 | Kenpaullone ≥98% | 10mg | $59 | 2021-12-16 | Buy |
| Arctom | AS025643 | Kenpaullone ≥98% | 50mg | $101 | 2021-12-16 | Buy |
Properties
Melting point :>300°C (dec.)
Boiling point :613.0±45.0 °C(Predicted)
Density :1.596±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 18 mg/mL, clear, yellow
pka :14.29±0.20(Predicted)
form :Yellow-brown solid
color :yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChIKey :QQUXFYAWXPMDOE-UHFFFAOYSA-N
CAS DataBase Reference :142273-20-9(CAS DataBase Reference)
Boiling point :613.0±45.0 °C(Predicted)
Density :1.596±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: 18 mg/mL, clear, yellow
pka :14.29±0.20(Predicted)
form :Yellow-brown solid
color :yellow
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.
InChIKey :QQUXFYAWXPMDOE-UHFFFAOYSA-N
CAS DataBase Reference :142273-20-9(CAS DataBase Reference)
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
Kenpaullone is an ATP-competitive inhibitor of several CDKs (cyclin-dependent kinases) as well as GSK-3β (glycogen synthase kinase 3β). It has been shown to inhibit GSK-3 with an IC50 value of 0.23 μM and CDK1/cyclin B, CDK2/cyclin A, CDK5/p25, and lymphocyte kinase with IC50 values of 0.4, 0.68, 0.85, and 0.47 μM, respectively. Due to the compound’s activity, Kenpaullone is useful in the study of cell cycle regulators. Kenpaullone is an inhibitor of cyclin E, ERK 2 and p35.Related product price
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Suppliers and manufacturers
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HANGZHOU CLAP TECHNOLOGY CO.,LTD
Zhejiang J&C Biological Technology Co.,Limited
