Glucagon Receptor Antagonist I
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- $74 - $583
- Product name: Glucagon Receptor Antagonist I
- CAS: 438618-32-7
- MF: C20H30N2OS
- MW: 346.53
- EINECS:
- MDL Number:MFCD01920208
- Synonyms:Glucagon Receptor Antagonist I;N-[3-cyano-6-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-ethylbutanamide;Butanamide, N-[3-cyano-6-(1,1-dimethylpropyl)-4,5,6,7-tetrahydrobenzo[b]thien-2-yl]-2-ethyl-;hGCGR Antagonist
5 prices
Selected condition：
Brand
- AK Scientific
- Cayman Chemical
Package
- 500μg
- 1mg
- 5mg
- ManufacturerAK Scientific
- Product number8227CC
- Product descriptionGlucagonReceptorAntagonistI
- Packaging5mg
- Price$583
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number8227CC
- Product descriptionGlucagonReceptorAntagonistI
- Packaging1mg
- Price$233
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number21223
- Product descriptionGlucagon Receptor Antagonist I ≥99%
- Packaging500μg
- Price$74
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21223
- Product descriptionGlucagon Receptor Antagonist I ≥99%
- Packaging1mg
- Price$132
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number21223
- Product descriptionGlucagon Receptor Antagonist I ≥99%
- Packaging5mg
- Price$476
- Updated2024-03-01
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 8227CC | GlucagonReceptorAntagonistI | 5mg | $583 | 2021-12-16 | Buy |
| AK Scientific | 8227CC | GlucagonReceptorAntagonistI | 1mg | $233 | 2021-12-16 | Buy |
| Cayman Chemical | 21223 | Glucagon Receptor Antagonist I ≥99% | 500μg | $74 | 2024-03-01 | Buy |
| Cayman Chemical | 21223 | Glucagon Receptor Antagonist I ≥99% | 1mg | $132 | 2024-03-01 | Buy |
| Cayman Chemical | 21223 | Glucagon Receptor Antagonist I ≥99% | 5mg | $476 | 2024-03-01 | Buy |
Properties
Boiling point :517.8±50.0 °C(Predicted)
Density :1.07±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO: soluble
form :White crystalline solid.
pka :13.46±0.40(Predicted)
Density :1.07±0.1 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO: soluble
form :White crystalline solid.
pka :13.46±0.40(Predicted)
Safety Information
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Description
Glucagon Receptor Antagonist I is a potent and selective cell-permeable thienyl-amide compound that acts as a competitive antagonist of the glucagon receptor. Exhibits binding to hGCGR with high affinity and prevents its interaction with glucagon (IC50 = 181 nM, KDB = 81 nM, and pA2 = 7.1 in membranes prepared from CHO-hGCGR). Also suppresses glucagon-induced glycogenolysis in human primary hepatocytes and in mice (50 mg/kg, ip).More related product prices
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