PAR-4 Agonist Peptide, amide TFA NEW
| Price | $47 | $147 | $247 |
| Package | 1mg | 5mg | 10mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2024-11-19 |
Product Details
| Product Name: PAR-4 Agonist Peptide, amide TFA | CAS No.: 1228078-65-6 |
| Purity: 100% | Supply Ability: 10g |
| Release date: 2024/11/19 |
Product Introduction
Bioactivity
| Name | PAR-4 Agonist Peptide, amide TFA |
| Description | PAR-4 Agonist Peptide, amide TFA (PAR-4-AP (TFA)), is a selective activator of the proteinase-activated receptor-4 (PAR-4) that does not affect PAR-1 or PAR-2, and its activity can be inhibited by a PAR-4 antagonist. |
| In vivo | SCID mice demonstrate a markedly enhanced abdominal response to colorectal distension (CRD), with distension levels ranging from 0.04 to 0.1 mL amplifying the intensity of the EMG response from 384% to 132%, respectively, as compared to BALB/cBy controls (P<0.01; P<0.01; P<0.01; P<0.001). Activation of PAR-4 significantly mitigates this hypersensitivity (P<0.01, P<0.05; P<0.05; P<0.05)[1]. |
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | H2O : 100 mg/mL (125.81 mM), Sonication is recommended. DMSO : 250 mg/mL (314.54 mM) |
| Keywords | Thrombin receptors | PAR4 Agonist Peptide, amide TFA | Protease Activated Receptor (PAR) | inhibit | PAR-4 Agonist Peptide, amide | Inhibitor | PAR-4-AP | PAR-4 Agonist Peptide, amide TFA | PAR 4 Agonist Peptide, amide TFA | AY-NH2 |
| Inhibitors Related | FSLLRY-NH2 TFA(245329-02-6 free base) | LRGILS-NH2 acetate | PAR-2 Activating Peptide acetate | Atopaxar | Vorapaxar sulfate | Trypsin | Vorapaxar | AY 77 | PAR-2-IN-1 | VKGILS-NH2 Acetate |
| Related Compound Libraries | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Peptide Compound Library | Inhibitor Library | NO PAINS Compound Library | Bioactive Compounds Library Max | GPCR Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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Recommended supplier
| Product name | Price | Suppliers | Update time | |
|---|---|---|---|---|
| $133.00/1mg |
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TargetMol Chemicals Inc.
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2024-11-19 | |
| $0.00/5mg |
VIP1Y
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TargetMol Chemicals Inc.
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| $30.00/1Box |
zhuzhou dingcheng meihei comestic co.,ltd
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2023-12-07 |
United States- Since: 2011-01-07
- Address: 36?Washington?Street, Wellesley?Hills
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