GPR40 agonist 6 NEW
Price | $53 |
Package | 2mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-19 |
Product Details
Product Name: GPR40 agonist 6 | CAS No.: 1798751-25-3 |
Supply Ability: 10g | Release date: 2024/11/19 |
Product Introduction
Bioactivity
Name | GPR40 agonist 6 |
Description | GPR40 agonist 6 (Compound 7a) is a potent and selective agonist of free fatty acid receptor 1 (FFAR1 or GPR40) with an EC50 of 0.058 μM against GPR40 [1]. |
In vitro | GPR40 agonist 6 (Compound 7a) exhibits an excellent ADME profile with negligible inhibition of key cytochrome P450 isoforms (1A2, 2C9, 2C19, 2D6, and 3A4) at 5 μM. It shows 98.6% human plasma protein binding, 404 μM aqueous solubility in PBS (pH 7.4), a microsomal stability half-life of 434 minutes in mice, and a Caco-2 permeability rate of 15.2 x 10^-6 cm/s, indicating promising pharmacokinetic properties. |
Storage | Shipping with blue ice. |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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- Since: 2011-01-07
- Address: 36?Washington?Street, Wellesley?Hills
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