Relugolix
- $32 - $3728.1
- Product name: Relugolix
- CAS: 737789-87-6
- MF: C29H27F2N7O5S
- MW: 623.63
- EINECS:237-099-7
- MDL Number:MFCD25976856
- Synonyms:TAK-385;TKA-385 Relugolix;TAK-385,Relugolix;CS-2851;TAK-385;TAK 385;TAK385;1-[4-[1-[(2,6-difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-methoxypyridazin-3-yl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-3-methoxyurea;10G,100G,500G,1KG;N-[4-[1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-1,2,3,4-tetrahydro-3-(6-methoxy-3-pyridazinyl)-2,4-dioxothieno[2,3-d]pyrimidin-6-yl]phenyl]-N'-methoxy urea
20 prices
Selected condition:
Brand
- AK Scientific
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
Package
- 1mg
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 250mg
- 1g
- ManufacturerAK Scientific
- Product number6863CR
- Product descriptionRelugolix
- Packaging10mg
- Price$370
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product number6863CR
- Product descriptionRelugolix
- Packaging25mg
- Price$691
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb573025
- Product descriptionRelugolix (TAK-385) >98%
- Packaging100mg
- Price$1133.9
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb573025
- Product descriptionRelugolix (TAK-385) >98%
- Packaging250mg
- Price$1802
- Updated2021-12-16
- Buy
- ManufacturerBiorbyt Ltd
- Product numberorb573025
- Product descriptionRelugolix (TAK-385) >98%
- Packaging1g
- Price$3728.1
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number29512
- Product descriptionTAK-385
- Packaging1mg
- Price$32
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29512
- Product descriptionTAK-385
- Packaging5mg
- Price$139
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29512
- Product descriptionTAK-385
- Packaging10mg
- Price$243
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number29512
- Product descriptionTAK-385
- Packaging25mg
- Price$533
- Updated2024-03-01
- Buy
- ManufacturerChemScene
- Product numberCS-5917
- Product descriptionRelugolix >98.0%
- Packaging1mg
- Price$70
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5917
- Product descriptionRelugolix >98.0%
- Packaging5mg
- Price$120
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5917
- Product descriptionRelugolix >98.0%
- Packaging10mg
- Price$190
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5917
- Product descriptionRelugolix >98.0%
- Packaging50mg
- Price$660
- Updated2021-12-16
- Buy
- ManufacturerChemScene
- Product numberCS-5917
- Product descriptionRelugolix >98.0%
- Packaging100mg
- Price$1100
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD11064717
- Product descriptionRelugolix(TAK385) 97%
- Packaging5mg
- Price$245
- Updated2021-12-16
- Buy
- ManufacturerCrysdot
- Product numberCD11064717
- Product descriptionRelugolix(TAK385) 97%
- Packaging10mg
- Price$350
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
AK Scientific | 6863CR | Relugolix | 10mg | $370 | 2021-12-16 | Buy |
AK Scientific | 6863CR | Relugolix | 25mg | $691 | 2021-12-16 | Buy |
Biorbyt Ltd | orb573025 | Relugolix (TAK-385) >98% | 100mg | $1133.9 | 2021-12-16 | Buy |
Biorbyt Ltd | orb573025 | Relugolix (TAK-385) >98% | 250mg | $1802 | 2021-12-16 | Buy |
Biorbyt Ltd | orb573025 | Relugolix (TAK-385) >98% | 1g | $3728.1 | 2021-12-16 | Buy |
Cayman Chemical | 29512 | TAK-385 | 1mg | $32 | 2024-03-01 | Buy |
Cayman Chemical | 29512 | TAK-385 | 5mg | $139 | 2024-03-01 | Buy |
Cayman Chemical | 29512 | TAK-385 | 10mg | $243 | 2024-03-01 | Buy |
Cayman Chemical | 29512 | TAK-385 | 25mg | $533 | 2024-03-01 | Buy |
ChemScene | CS-5917 | Relugolix >98.0% | 1mg | $70 | 2021-12-16 | Buy |
ChemScene | CS-5917 | Relugolix >98.0% | 5mg | $120 | 2021-12-16 | Buy |
ChemScene | CS-5917 | Relugolix >98.0% | 10mg | $190 | 2021-12-16 | Buy |
ChemScene | CS-5917 | Relugolix >98.0% | 50mg | $660 | 2021-12-16 | Buy |
ChemScene | CS-5917 | Relugolix >98.0% | 100mg | $1100 | 2021-12-16 | Buy |
Crysdot | CD11064717 | Relugolix(TAK385) 97% | 5mg | $245 | 2021-12-16 | Buy |
Crysdot | CD11064717 | Relugolix(TAK385) 97% | 10mg | $350 | 2021-12-16 | Buy |
Properties
Melting point :228 °C (decomp)(Solv: ethyl acetate (141-78-6); tetrahydrofuran (109-99-9))
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O
Density :1.442±0.06 g/cm3(Predicted)
storage temp. :Store at -20°C
solubility :DMSO:20.0(Max Conc. mg/mL);32.1(Max Conc. mM)
Ethanol:1.0(Max Conc. mg/mL);1.6(Max Conc. mM) form :A crystalline solid
pka :13.17±0.70(Predicted)
color :White to off-white
InChIKey :AOMXMOCNKJTRQP-UHFFFAOYSA-N
SMILES :N(C1=CC=C(C2SC3=C(C=2CN(C)C)C(=O)N(C2=NN=C(OC)C=C2)C(=O)N3CC2=C(F)C=CC=C2F)C=C1)C(NOC)=O
Safety Information
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Signal word: | Warning | ||||||||||||||||||||||
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Description
Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. It possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209). Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al.More related product prices
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