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FGTI-2734

FGTI-2734 ??? ???
?? ??:
1247018-19-4
???:
FGTI-2734
???(??):
FGTI-2734;FGTI-2734, 10 mM in DMSO;2-Pyridinesulfonamide, N-[2-[(4-cyano-2-fluorophenyl)[(1-methyl-1H-imidazol-5-yl)methyl]amino]ethyl]-N-(cyclohexylmethyl)-;pancreatic,patient-derived,geranylgeranyl,farnesyl,inhibit,Farnesyl Transferase,mimetic,FGTI2734,Inhibitor,membrane,Ftase,FGTI-2734,KRAS,FGTI 2734,C-terminal,transferase,tumors,localization
CBNumber:
CB75540586
???:
C26H31FN6O2S
??? ??:
510.63
MOL ??:
1247018-19-4.mol

FGTI-2734 ??

?? ?
770.1±70.0 °C(Predicted)
??
1.28±0.1 g/cm3(Predicted)
?? ??
Store at -20°C
???
DMSO:50.0(Max Conc. mg/mL);97.92(Max Conc. mM)
??? ??
Solid
?? ?? (pKa)
6.60±0.10(Predicted)
??
White to off-white

??

FGTI-2734 C??? ??, ??, ??

FGTI-2734 ?? ?? ? ???

???

?? ??


FGTI-2734 ?? ??

???( 28)?? ??
??? ?? ??? ?? ?? ? ??
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