PROXYFAN MALEATE Chemische Eigenschaften,Einsatz,Produktion Methoden
Biologische Aktivit?t
High affinity histamine H 3 receptor ligand (pK i = 8.62) that acts as a protean agonist at recombinant and native receptors. In functional studies, activity ranges from full agonist to inverse agonist depending on system used. Displays partial agonist effects on cAMP inhibition and MAPK activity, neutral antagonist activity on histamine release and partial inverse agonism of [ 3 H]-arachidonic acid release.
PROXYFAN MALEATE Upstream-Materialien And Downstream Produkte
Upstream-Materialien
Downstream Produkte