K-252C
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- CAS-Nr.
- 85753-43-1
- Englisch Name:
- K-252C
- Synonyma:
- K-252C;Staurosporonine;Staurosporinone;STAUROSPORINE AGLYCONE;K-252c(Staurosporinone);Staurosporinone, K-252c;K252c, Ready Made Solution;Staurosporine Aglycone >99%;K-252c - CAS 85753-43-1 - Calbiochem;Staurosporinone, Staurosporine Aglycone
- CBNumber:
- CB3406463
- Summenformel:
- C20H13N3O
- Molgewicht:
- 311.34
- MOL-Datei:
- 85753-43-1.mol
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K-252C Eigenschaften
- Schmelzpunkt:
- >200°C (dec.)
- storage temp.
- −20°C
- L?slichkeit
- DMSO: 10 mg/mL, soluble
- Aggregatzustand
- solid
- Farbe
- Pale Brown to Light Brown
- Wasserl?slichkeit
- Soluble in DMSO at 25mM. Also soluble in methanol. Insoluble in water.
K-252C Chemische Eigenschaften,Einsatz,Produktion Methoden
S-S?tze Betriebsanweisung:
S22:Staub nicht einatmen.
S24/25:Berührung mit den Augen und der Haut vermeiden.
Verwenden
Inhibits protein kinase C
Biologische Aktivit?t
Inhibitor of protein kinase C (IC 50 = 2.45 μ M) that displays ~ 10-fold selectivity over protein kinase A (IC 50 = 25.7 μ M). Also inhibits β -lactamase, malate dehydrogenase and chymotrypsin (IC 50 values are 8, 8 and 10 μ M respectively). Exhibits antiviral activity against GCV-sensitive and -resistant strains of human cytomegalovirus (HCMV) (IC 50 values range from 0.13-0.32 μ M). Shows no activity against herpes simplex virus (HSV).
K-252C Upstream-Materialien And Downstream Produkte
Upstream-Materialien
Downstream Produkte
K-252C Anbieter Lieferant Produzent Hersteller Vertrieb H?ndler.
Global( 87)Lieferanten
85753-43-1()Verwandte Suche:
Kaliumnitrat
(+)-2,3,10,11,12,13-Hexahydro-10-methoxy-9-methyl-11-(methylamino)-9,13-epoxy-1H,9H-diindolo (1,2,3-gh: 3'2',1'-1m)pyrrolo(3,4-j)-(1,7)benzodiazonin-1-on, (9 alpha,10 beta, 11 beta, 13 alpha)-
3,4-Dihydroisochinolin
(Maleato)trioxotetrablei
Schwefelsaeurediamid
Kaliumabietat
- K-252C
- STAUROSPORINE AGLYCONE
- Staurosporinone
- 6,7,12,13-Tetrahydro-5H-indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one
- Staurosporine Aglycone >99%
- Staurosporinone, K-252c
- K-252c(Staurosporinone)
- K252c / Staurosporine Aglycone>99%/ Staurosporinone, K-252C /
6,7,12,13-Tetrahydro-5H-Indolo[2,3-A]Pyrrolo[3,4-C]Carbazol-5-One
- K252c, Ready Made Solution
- Staurosporonine
- Staurosporinone, Staurosporine Aglycone
- K-252c - CAS 85753-43-1 - Calbiochem
- 5H-Indolo[2,3-a]pyrrolo[3,4-c]carbazol-5-one, 6,7,12,13-tetrahydro-
- 85753-43-1
- C20H13N3O
- v-Src Sarcoma (Schmidt-Ruppin A-2) Viral Oncogene Homolog (Src)
- Kinase/Phosphatase Biology
- Non-Receptor Tyrosine Kinase Inhibitors
- BioChemical
- Cell Biology
- Cell Signaling and Neuroscience
- Inhibitor
