H-D-PHG-OME HCL synthesis
- Product Name:H-D-PHG-OME HCL
- CAS Number:19883-41-1
- Molecular formula:C9H12ClNO2
- Molecular Weight:201.65
Yield:19883-41-1 98.9%
Reaction Conditions:
with dichlorosulfoxide at 0 - 75; for 2 h;
Steps:
First step
General procedure: The methyl-esterification reaction of L-phenylalanine.To a suspension of L-phenylalanine (1 g, 6.05 mmol, 1.0 equiv) inmethanol (25 mL) cooled to 0 C was added thionyl chloride(475 mL, 6.66 mmol, 1.5 equiv) slowly. After 10 min, the reactionmixture was heated to 75 C to reflux for 2 h. After completion(monitored by TLC), the solvent was removed in vacuo, and at thistime, a white solid was formed methyl L-phenylalaninate hydrochloride(1.23 g, quantitative yield).
References:
Liu, Sha;Jing, Li;Yu, Zhu-Jun;Wu, Chengyong;Zheng, Yongxiang;Zhang, En;Chen, Qiang;Yu, Yamei;Guo, Li;Wu, Yong;Li, Guo-Bo [European Journal of Medicinal Chemistry,2018,vol. 145,p. 649 - 660]
98-80-6
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$5.00/5g
19883-41-1
342 suppliers
$6.00/5g
67-56-1
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$9.00/25ml
33125-05-2
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19883-41-1
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15028-40-7
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15028-39-4
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19883-41-1
342 suppliers
$6.00/5g
67-56-1
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$9.00/25ml
875-74-1
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15028-39-4
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$5.00/1g
19883-41-1
342 suppliers
$6.00/5g