5-BROMO-2-(2,2,2-TRIFLUORO-ETHOXY)-PYRIMIDINE synthesis
- Product Name:5-BROMO-2-(2,2,2-TRIFLUORO-ETHOXY)-PYRIMIDINE
- CAS Number:433683-47-7
- Molecular formula:C6H4BrF3N2O
- Molecular Weight:257.01
6226-25-1
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38353-06-9
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433683-47-7
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Yield:433683-47-7 296 mg
Reaction Conditions:
with caesium carbonate in N,N-dimethyl-formamide at 80; for 2 h;
Steps:
3.B B) 5-bromo-2-(2,2,2-trifluoroethoxy)pyrimidine
A mixture of 5-bromopyrimidin-2-ol (500 mg), 2,2,2-trifluoroethyl trifluoromethanesulfonate (796 mg), cesium carbonate (1397 mg) and DMF (5 mL) was stirred at 80° C. for 2 hr.
Water was added to the mixture and the mixture was extracted with ethyl acetate.
The organic layer was separated, washed with saturated brine, dried over anhydrous magnesium sulfate and concentrated under reduced pressure.
The residue was purified by silica gel column chromatography (ethyl acetate/hexane) to give the title compound (296 mg).
1H NMR (300 MHz, CDCl3) 54.79 (2H, q, J=8.2 Hz), 8.58 (2H, s).
References:
US2020/39957,2020,A1 Location in patent:Paragraph 0641
75-89-8
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32779-36-5
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433683-47-7
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$50.00/250mg
855719-15-2
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38275-48-8
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$16.00/250mg
433683-47-7
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$50.00/250mg
75-89-8
474 suppliers
$9.00/1g
32779-37-6
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$9.00/1g
433683-47-7
31 suppliers
$50.00/250mg
75-89-8
474 suppliers
$9.00/1g
62802-38-4
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433683-47-7
31 suppliers
$50.00/250mg