5-bromo-N-(4,4,5,5-tetradeuterio-1H-imidazol-2-yl)quinoxalin-6-amine
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- $93 - $775
- Product name: 5-bromo-N-(4,4,5,5-tetradeuterio-1H-imidazol-2-yl)quinoxalin-6-amine
- CAS: 1184971-51-4
- MF: C11H10BrN5
- MW: 292.14
- EINECS:
- MDL Number:
- Synonyms:5-bromo-N-(4,4,5,5-tetradeuterio-1H-imidazol-2-yl)quinoxalin-6-amine;5-bromo-N-(4,5-dihydro-1H-imidazol-2-yl-4,4,5,5-d4)quinoxalin-6-amine
4 prices
Selected condition：
Brand
- AK Scientific
- Cayman Chemical
Package
- 500μg
- 1mg
- 5mg
- ManufacturerAK Scientific
- Product number5496DF
- Product description5-Bromo-N-(4,4,5,5-tetradeuterio-1H-imidazol-2-yl)quinoxalin-6-amine
- Packaging1mg
- Price$299
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number25465
- Product descriptionBrimonidine-d4 ≥99% deuterated forms (d1-d4)
- Packaging500μg
- Price$93
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number25465
- Product descriptionBrimonidine-d4 ≥99% deuterated forms (d1-d4)
- Packaging1mg
- Price$176
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number25465
- Product descriptionBrimonidine-d4 ≥99% deuterated forms (d1-d4)
- Packaging5mg
- Price$775
- Updated2024-03-01
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | 5496DF | 5-Bromo-N-(4,4,5,5-tetradeuterio-1H-imidazol-2-yl)quinoxalin-6-amine | 1mg | $299 | 2021-12-16 | Buy |
| Cayman Chemical | 25465 | Brimonidine-d4 ≥99% deuterated forms (d1-d4) | 500μg | $93 | 2024-03-01 | Buy |
| Cayman Chemical | 25465 | Brimonidine-d4 ≥99% deuterated forms (d1-d4) | 1mg | $176 | 2024-03-01 | Buy |
| Cayman Chemical | 25465 | Brimonidine-d4 ≥99% deuterated forms (d1-d4) | 5mg | $775 | 2024-03-01 | Buy |
Properties
storage temp. :Store at -20°C
solubility :DMSO: soluble; Water: 1.5 mg/ml
form :A solid
solubility :DMSO: soluble; Water: 1.5 mg/ml
form :A solid
Safety Information
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Description
Brimonidine-d4 is intended for use as an internal standard for the quantification of brimonidine by GC- or LC-MS. Brimonidine is an agonist of α2-adrenergic receptors (α2-ARs; Kis = 2.7, 52, and 44 nM for α2A, α2B, and α2C-ARs, respectively, in CHO cells).1 It is selective for α2-ARs over α1-ARs (Ki = 1,800 nM in human brain). Brimonidine lowers intraocular pressure in DBA/2J mice, a model of glaucoma, to control levels when applied topically to the eye as a 0.1% solution.2 It also inhibits glutamate release, prevents upregulation of NMDA receptors containing NR1 and NR2A subunits, and protects rat retinal ganglion cells against glutamate excitotoxicity in a rat model of retinal ischemia when administered at a dose of 1 mg/kg per day.3 Formulations containing brimonidine have been used in the treatment of open-angle glaucoma and ocular hypertension.More related product prices
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$185-460 - N-(4,5-Dihydro-1H-iMidazol-2-yl)-6-quinoxalinaMine
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$5-3500