中文名：VUF 10166,5-HT3拮抗劑

英文名：VUF 10166

中文別名：2-氯-3-(4-甲基-1-哌嗪基)喹喔啉

英文別名：155584-74-0|2-chloro-3-(4-methylpiperazin-1-yl)quinoxaline|VUF 10166|Quinoxaline, 2-chloro-3-(4-methyl-1-piperazinyl)-|CHEMBL261010|VUF10166|VUF10166;VUF-10166|2-Chloro-3-(4-methyl-1-piperazinyl)quinoxaline|SCHEMBL404203|DTXSID60640663|HMS3651F21|HMS3884N

純度：≥99%

貨號：V129763

包裝：10mg、50mg、250mg

Cas號：155584-74-0

存儲溫度：-20°C儲存

產品介紹：

VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower. VUF10166 shows low activity to 5-HT3AB receptor with Ki of 22 nM. VUF10166 may be used to can distinguish between 5-HT3A and 5-HT3AB receptors. VUF10166 has no activity to α7 nACh receptor. VUF10166 also acts as a partial agonist at 5-HT3A receptors with EC50 of 5.2 μM, which shows that VUF10166 is unlikely to bind in the receptor pore.

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