4 | 2183239-01-0 | CP 526555-d4 | 伐尼克蘭-d4 | Isotope-Labeled Compounds | nAChR | Nicotinic acetylcholine receptors | Inhibitor | inhibitor | inhibit"/>

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  2. Others Membrane Transporter/Ion Channel Neuronal Signaling
  3. Isotope-Labeled Compounds nAChR
  4. Varenicline-d4

Varenicline-d4  (Synonyms: 伐尼克蘭-d4; CP 526555-d4)

目錄號(hào): HY-10019S
產(chǎn)品使用指南

Varenicline-d4 是 Varenicline 氘代物。Varenicline (CP 526555) 是 α4β2 nAChR 煙堿乙酰膽堿受體的部分激動(dòng)劑 (EC50=2.3 μM)。Varenicline 是 α3β4 nAChR 和 α7 nAChR 乙酰膽堿受體完全激動(dòng)劑，EC50 值分別為 55 μM 和 18 μM。Varenicline 是一種基于胞嘧啶結(jié)構(gòu)的煙堿配體，有潛力用于戒煙方面的研究。

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Varenicline-d<sub>4</sub> Chemical Structure

Varenicline-d4 Chemical Structure

CAS No. : 2183239-01-0

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規(guī)格 價(jià)格 是否有貨 數(shù)量
500 μg ￥1962
3 - 4 周
1 mg 詢(xún)價(jià)
5 mg 詢(xún)價(jià)

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Customer Review

Other Forms of Varenicline-d4:

  • 生物活性

  • 純度 & 產(chǎn)品資料

  • 參考文獻(xiàn)

生物活性

Varenicline-d4 is deuterium labeled Varenicline. Varenicline (CP 526555) is a potent partial agonist for α4β2 nicotinic acetylcholine receptor (nAChR) with an EC50 value of 2.3 μM. Varenicline is a full agonist for α3β4 and α7 nAChRs with EC50 values of 55 μM and 18 μM, respectively[1]. Varenicline is a nicotinic ligand based on the structure of cytisine, has the potential for smoking cessation treatment[2].

體外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

215.29

Formula

C13H9D4N3
CAS 號(hào)
非標(biāo)記 CAS
中文名稱(chēng)

伐尼克蘭-d4
運(yùn)輸條件

Room temperature in continental US; may vary elsewhere.
儲(chǔ)存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
純度 & 產(chǎn)品資料
參考文獻(xiàn)

  • 摩爾計(jì)算器

  • 稀釋計(jì)算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

質(zhì)量   濃度   體積   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

濃度 (start) × 體積 (start) = 濃度 (final) × 體積 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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產(chǎn)品名稱(chēng)：
Varenicline-d4
目錄號(hào)：
HY-10019S
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