SB 207499 - Cilomilast | Ariflo

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1592

CAS [153259-65-5]

MF C20H25NO4
MW 343.42

Purity: 99%
Soluble in 0.1N NaOH(aq) and DMSO

SB 207499

Description

Selective and orally active inhibitor of phosphodiesterase-4 (PDE4); a potential agent for the treatment of respiratory disorders such as asthma and Chronic Obstructive Pulmonary Disease (COPD); a second generation PDE4 inhibitor, reduces tumor necrosis factor α and interleukin-4 production in vivo

TJ Torphy et al. Ariflo (SB 207499), a second generation phosphodiesterase 4 inhibitor for the treatment of asthma and COPD: from concept to clinic. Pulmonary Pharmacol. Ther. 1999, 12(2), 131-135.

H Ochiai et al. Highly potent PDE4 inhibitors with therapeutic potential. Bioorg. Med. Chem. Lett. 2004, 14(1), 207-210.

SB Christensen et al. 1,4-Cyclohexanecarboxylates: Potent and Selective Inhibitors of Phosophodiesterase 4 for the Treatment of Asthma. J. Med. Chem. 1998, 41(6), 821.

DE Griswold etal. SB 207499 (Ariflo), a Second Generation Phosphodiesterase 4 Inhibitor, Reduces Tumor Necrosis Factor α and Interleukin-4 Production in vivo.
J. Pharmacol. Exp. Ther. 1998, 287(2), 705-711.

Cell Signaling & Oncology CNS Pain & Inflammation EC 3.1.4.53 PDE

PDE4 inhibitor

Chemical name

4-Cyano-4-(3-(cyclopentyloxy)-4-methoxyphenyl)cyclohexanecarboxylic acid

Parent CAS No.

[153259-65-5]

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Size	Unit Price	Stock
5 mg	€70.00	In Stock
25 mg	€220.00	In Stock

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Size	Unit Price	Stock
2 x 5 mg	€100.00	In Stock
2 x 25 mg	€340.00	In Stock

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天堂网亚洲,天天操天天搞,91视频高清,菠萝蜜视频在线观看入口,美女视频性感美女视频,95丝袜美女视频国产,超高清美女视频图片

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SB 207499 - Cilomilast | Ariflo

Description

Chemical name

Parent CAS No.

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