Phenyltoloxamine NEW
Price | $1520 | $1980 | $2500 |
Package | 25mg | 50mg | 100mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-19 |
Product Details
Product Name: Phenyltoloxamine | CAS No.: 92-12-6 |
Supply Ability: 10g | Release date: 2024/11/19 |
Product Introduction
Bioactivity
Name | Phenyltoloxamine |
Description | Phenyltoloxamine (Bistrimin) is an antihistamine with sedative and analgesic properties, and it exhibits strong Sigma-1 receptor binding affinity with a Ki of 160 nM [1] [2] [3]. |
In vitro | Phenyltoloxamine, within a concentration range of 10-50 μM over 24 hours, demonstrates cytotoxic effects on EVSA-T cells [2]. Additionally, it exhibits significant binding affinity for the Sigma 1 Receptor (S1R), with a K i value of 160 nM [3]. At a higher concentration of 100 μM, Phenyltoloxamine inhibits the CYP2D6 enzyme in human liver by 99.0% [4]. |
Storage | Shipping with blue ice. |
Company Profile Introduction
TargetMol Chemicals Inc. is headquartered in Boston, MA, and specializes in products and services that serve the research needs of chemical and biological scientists worldwide. With a client base in 40+ countries, TargetMol has evolved into one of the biggest global research suppliers for compound libraries and small molecule compounds.
170+ Compound Libraries, 10000+ Noval Small Molecucles,16000+ Nature Compounds
TargetMol diligently updates and offers over 170 types of compound libraries and a wide range of high-quality research chemicals, including inhibitors, activators, natural products, peptides, antibodies , and novel life-science kits for laboratory and scientific use. In addition, our lab allows us to conduct CADD (computer-aided drug design) and chemical synthesis to meet the customization needs of our clients.
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- Since: 2011-01-07
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