L-368,899 hydrochloride NEW
Price | $113 | $158 | $255 |
Package | 2mg | 5mg | 10mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-12 |
Product Details
Product Name: L-368,899 hydrochloride | CAS No.: 160312-62-9 |
Purity: 99.59% | Supply Ability: 10g |
Release date: 2024/11/12 |
Product Introduction
Bioactivity
名稱 | L-368,899 hydrochloride |
描述 | L-368,899 hydrochloride is an orally available and selective nonpeptide oxytocin receptor (OXTR) antagonist for the prevention of preterm labor.L-368,899 hydrochloride prevents oxytocin-induced anti-anomalous pain and anti-nausea, and may be useful for the study of depression. |
體外活性 | L-368,899 hydrochloride is an effective non-peptide oxytocin receptor antagonist, with IC50 values of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptors, respectively[1]. |
體內(nèi)活性 | L-368,899 (5 mg/kg; oral administration) has oral bioavailabilities of 14% and 18% in female and male rats, respectively[2]. |
存儲條件 | store at low temperature,keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度 | H2O : 2 mg/mL (3.38 mM), Sonication is recommended. DMSO : 100 mg/mL (169.14 mM), Sonication is recommended. |
關鍵字 | L-368,899 Hydrochloride | L368,899 hydrochloride | L 368,899 hydrochloride |
相關產(chǎn)品 | YNT-185 | Orexin 2 Receptor Agonist | IPSU | MK-3697 | Filorexant | DORA-22 | Orexin B, rat, mouse Acetate | OXA (17-33) acetate | PF3274167 | ACT-462206 | Seltorexant | TCS 1102 |
相關庫 | 經(jīng)典已知活性庫 | 神經(jīng)信號分子庫 | 抑制劑庫 | 口服活性化合物庫 | 已知活性化合物庫 | GPCR靶點分子庫 |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
You may like
Recommended supplier
Product name | Price | Suppliers | Update time | |
---|---|---|---|---|
$45.00/1kg |
VIP1Y
|
Hebei Zhuanglai Chemical Trading Co Ltd
|
2024-12-03 | |
$10.00/1kg |
VIP1Y
|
Hebei Zhuanglai Chemical Trading Co.,Ltd
|
2024-05-31 | |
$20.00/1kg |
VIP2Y
|
Hebei Miaoyin Technology Co.,Ltd
|
2023-04-06 | |
$113.00/2mg |
VIP5Y
|
TargetMol Chemicals Inc.
|
2024-11-12 |
- Since: 2011-01-07
- Address: 36?Washington?Street, Wellesley?Hills
INQUIRY