Estradiol 3-sulfamate NEW
Price | $147 | $297 | $476 |
Package | 1mg | 5mg | 10mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-20 |
Product Details
Product Name: Estradiol 3-sulfamate | CAS No.: 172377-52-5 |
Purity: 96.68% | Supply Ability: 10g |
Release date: 2024/11/20 |
Product Introduction
Bioactivity
Name | Estradiol 3-sulfamate |
Description | Estradiol 3-sulfamate (BLE 00084) is an orally active and highly potent steroidal estrone sulfatase (ES) inhibitor.Estradiol 3-sulfamate has a K(i) value of 73 nM for ES in human placental microsomes and can be used in the study of breast cancer. |
In vitro | Compared to the lead compound EMATE, Estradiol 3-sulfamate exhibits superior inhibitory activity against estrone sulfatase[1]. |
In vivo | Estradiol 3-sulfamate readily transforms into its metabolite EMATE in the gut, making it a more effective STS inhibitor[2]. |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO : 50 mg/mL (142.26 mM), Sonication is recommended. |
Keywords | Estradiol 3sulfamate | Estradiol 3-sulfamate | ES-J-995 | ES-J995 | BLE00084 | BLE-00084 | Estradiol 3 sulfamate |
Inhibitors Related | Kaempferol | Tamoxifen | Estradiol | Estradiol benzoate | ARV-471 | Cholesterol | Estriol | Chrysin | Ethisterone | Estrone |
Related Compound Libraries | Bioactive Compound Library | Bioactive Compounds Library Max |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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- Since: 2011-01-07
- Address: 36?Washington?Street, Wellesley?Hills
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