D3-βArr NEW
Price | $40 | $68 | $147 |
Package | 5mg | 10mg | 25mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-17 |
Product Details
Product Name: D3-βArr | CAS No.: 662164-09-2 |
Purity: 98.82% | Supply Ability: 10g |
Release date: 2024/11/17 |
Product Introduction
Bioactivity
名稱 | D3-βArr |
描述 | D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct TSHR activation. |
體外活性 | D3-βArr stimulated β-Arr 1 translocation with an efficacy threefold greater than TSH. The EC50 for β-Arr 1 translocation by D3-βArr was 11.6 μM. D3-βArr (10 μM) increased the efficacy of TSH in the translocation of β-Arr 1 at a maximum of 5.1-fold over TSH alone. |
存儲(chǔ)條件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度 | DMSO : 100 mg/mL (299.91 mM) |
關(guān)鍵字 | Thyroid-stimulating hormone Receptor | D3-bArr | Thyrotropin receptor | inhibit | D3-βArr | D3-betaArr | D3βArr | TSH Receptor | Inhibitor | D-3-βArr | NCGC 00379308 | NCGC-00379308 | D3 βArr |
相關(guān)產(chǎn)品 | Teprotumumab | TSHR antagonist S37 | ML224 | VA-K-14 hydrochloride | Org41841 | ML-109 | NCGC00229600 |
相關(guān)庫(kù) | 成骨分子庫(kù) | 核受體化合物庫(kù) | 經(jīng)典已知活性庫(kù) | 膜蛋白靶向化合物庫(kù) | NO PAINS 化合物庫(kù) | 已知活性化合物庫(kù) | GPCR靶點(diǎn)分子庫(kù) |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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