AR-C155858 NEW
Price | $97 | $297 | $517 |
Package | 1mg | 5mg | 10mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-19 |
Product Details
Product Name: AR-C155858 | CAS No.: 496791-37-8 |
Purity: 98.84% | Supply Ability: 10g |
Release date: 2024/11/19 |
Product Introduction
Bioactivity
Name | AR-C155858 |
Description | AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM). |
In vitro | AR-C155858, at concentrations ranging from 10 nM to 100 nM, effectively inhibits the activity of MCT1/MCT2 C-terminal chimeras[1]. This compound also demonstrates time- and concentration-dependent inhibition of MCT1 when expressed in Xenopus oocytes[2]. Furthermore, AR-C155858 exhibits an inhibitory effect on MCT2, achieving 70% inhibition at 10 nM, with inhibition levels increasing gradually, indicative of a dissociation constant (Ki) value significantly lower than 10 nM. |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO : 40 mg/mL (86.67 mM) |
Keywords | inhibit | Inhibitor | AR-C-155858 | AR-C 155858 | Monocarboxylate Transporter | AR-C155858 | ARC155858 | AR C155858 |
Inhibitors Related | 7ACC1 | BAY-8002 | AZD0095 | MCT1-IN-3 | Niflumic acid | D-Phenylalanine | AZD3965 | MSC-4381 | α-Cyano-4-hydroxycinnamic acid | 7ACC2 | Lactate transportor 1 | VB124 |
Related Compound Libraries | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Inhibitor Library | NO PAINS Compound Library | Bioactive Compounds Library Max | Ion Channel Targeted Library | Anti-Cancer Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
You may like
Recommended supplier
Product name | Price | Suppliers | Update time | |
---|---|---|---|---|
$2580.00/50mg |
VIP1Y
|
TargetMol Chemicals Inc.
|
2024-10-28 | |
$653.00/5mg |
VIP3Y
|
TargetMol Chemicals Inc.
|
2024-10-28 | |
$1.00/1KG |
VIP6Y
|
Hebei Weibang Biotechnology Co., Ltd
|
2024-10-28 | |
$97.00/1mg |
VIP3Y
|
TargetMol Chemicals Inc.
|
2024-11-19 |
- Since: 2011-01-07
- Address: 36?Washington?Street, Wellesley?Hills
INQUIRY