TLX agonist 1
|
|
|
- CAS號:
- 958323-31-4
- 英文名:
- TLX agonist 1
- 英文別名:
- CCRP2;TLX a onist 1;TLX agonist 1;TLX agonist 1, 10 mM in DMSO;(4-Benzhydrylpiperazin-1-yl)(1,5-dimethyl-1H-pyrazol-3-yl)methanone;Methanone, (1,5-dimethyl-1H-pyrazol-3-yl)[4-(diphenylmethyl)-1-piperazinyl]-;TLX agonist-1,transcriptional,TLX agonist 1,repressive,Inhibitor,ligand,inhibit,TLX agonist1,orphan
- 中文名:
- TLX agonist 1
- 中文別名:
- TLX激動劑1;化合物TLX AGONIST 1;化合物TLX AGONIST 1,10 MM DMSO 溶液;(4-苯甲?；哙?1-基)(1,5-二甲基-1H-吡唑-3-基)甲酮
- CBNumber:
- CB35832809
- 分子式:
- C23H26N4O
- 分子量:
- 374.48
- MOL File:
- 958323-31-4.mol
|
|
|
TLX agonist 1化學(xué)性質(zhì)
-
沸點:
-
539.6±50.0 °C(Predicted)
-
|
-
密度:
-
1.16±0.1 g/cm3(Predicted)
-
|
-
儲存條件:
-
2-8°C
-
|
-
溶解度:
-
DMSO: 62.5 mg/mL (166.90 mM)
-
|
-
酸度系數(shù)(pKa):
-
5.78±0.10(Predicted)
-
|
-
形態(tài):
-
Solid
-
|
-
顏色:
-
White to off-white
-
|
TLX agonist 1性質(zhì)、用途與生產(chǎn)工藝
TLX agonist 1 (CCRP2, SUN23314) 是一種 orphan nuclear receptor tailless (TLX, NR2E1) 的調(diào)節(jié)劑，其EC50值為1.0 μM，Kd值為650 nM。TLX agonist 1 (CCRP2, SUN23314) 與重組TLX蛋白結(jié)合并增強TLX轉(zhuǎn)錄抑制活性。
| Target | Value |
NR2E1
(Cell-free assay)
|
650 nM(Kd)
|
NR2E1
(Cell-free assay)
|
1.0 μM(EC50)
|
TLX agonist 1
上下游產(chǎn)品信息
上游原料
下游產(chǎn)品
| 更新日期 | 產(chǎn)品編號 | 產(chǎn)品名稱 | CAS編號 | 包裝 | 價格 |
|---|
| 2025/05/22 | HY-135572 | TLX agonist 1
TLX agonist 1 | 958323-31-4 | 1mg | 500元 |
| 2025/05/22 | HY-135572 | TLX agonist 1
TLX agonist 1 | 958323-31-4 | 5mg | 1100元 |
958323-31-4, TLX agonist 1 相關(guān)搜索:
- 藥靶配體
- 抑制劑
- 化合物TLX AGONIST 1,10 MM DMSO 溶液
- TLX激動劑1
- 化合物TLX AGONIST 1
- (4-苯甲?；哙?1-基)(1,5-二甲基-1H-吡唑-3-基)甲酮
- 958323-31-4
- TLX agonist 1, 10 mM in DMSO
- TLX a onist 1
- TLX agonist-1,transcriptional,TLX agonist 1,repressive,Inhibitor,ligand,inhibit,TLX agonist1,orphan
- CCRP2
- (4-Benzhydrylpiperazin-1-yl)(1,5-dimethyl-1H-pyrazol-3-yl)methanone
- Methanone, (1,5-dimethyl-1H-pyrazol-3-yl)[4-(diphenylmethyl)-1-piperazinyl]-
- TLX agonist 1