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951322-11-5

中文名稱 DEFORMYLFLUSTRABROMINE HYDROCHLORIDE
英文名稱 dFBr hydrochloride
CAS 951322-11-5
分子式 C16H21BrN2*ClH
分子量 357.72
MOL 文件 951322-11-5.mol
951322-11-5 結(jié)構(gòu)式 951322-11-5 結(jié)構(gòu)式

基本信息

中文別名
化合物 T11004
英文別名
dFBr hydrochloride
Deformylflustrabromine hydrochloride
6-Bromo-2-(1,1-dimethyl-2-propen-1-yl)-N-methyl-1H-indole-3-ethanamine hydrochloride

物理化學(xué)性質(zhì)

儲存條件2-8°C
溶解度二甲基亞砜:≥10mg/mL
形態(tài)粉末
顏色白色至米色

安全數(shù)據(jù)

WGK Germany3

常見問題列表

生物活性
Desformylflustrabromine hydrochloride 是一個有選擇性的 α4β2 神經(jīng)元煙堿乙酰膽堿受體 (nAChR) 激動劑,其 pEC50 值為 6.48。
靶點

α 4 β 2 nAChR

體外研究

Desformylflustrabromine hydrochloride is a selective agonist of α 4 β 2 neuronal nicotinic acetylcholine receptor (nAChR) with a pEC 50 of 6.48. ACh-induced currents are potentiated and inhibited by Desformylflustrabromine hydrochloride in the high sensitivity (HS) and low sensitivity (LS) isoform preparations, although Desformylflustrabromine hydrochloride displays a higher potency on the LS isoform (pEC 50 =6.4±0.2) compare with the HS isoform (pEC 50 =5.6±0.2). Desformylflustrabromine hydrochloride potentiates ACh-induced responses of wild-type receptors expressed using the HS isoform preparation maximally by 350±20%, which is similar to receptors expressed via the LS isoform preparation (350±30%).

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