| Identification | Back Directory | [Name]
CETP-IN-3 | [CAS]
939391-31-8 | [Synonyms]
CETP-IN-3
CETP IN 3,CETPIN3
CETP-IN-3 (COMPOUND 13) | [Molecular Formula]
C30H24F12N2O4 | [MDL Number]
MFCD32174284 | [MOL File]
939391-31-8.mol | [Molecular Weight]
704.5 |
| Hazard Information | Back Directory | [Description]
CETP-IN-3 (Compound 13) is an small molecule inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP. CETP-IN-3 for the CETP inhibitory activity in the scintillation proximity (SPA) and whole plasma assay (WPA) with IC50s of 0.002 μM and 0.06 μM, respectively[1].
| [References]
[1]. Finlay HJ, et al. Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor. ACS Med Chem Lett. 2019 May 6; 10(6):911-916. |
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