Identification | Back Directory | [Name]
(E)-(4R,9aS)-7-[3-Methoxy-4-(4-methyl-1H-imidazol-1-yl)benzylidene]-4-(3,4,5-trifluorophenyl)hexahydropyrido[2,1-c][1,4]oxazin-6-one | [CAS]
937812-80-1 | [Synonyms]
HYR-141 Otamixaban SynonyMs: HYR-141 γ-Secretase Modulators γ-Secretase Modulators gaMMa-Secretase Modulators AMyloid-β production inhibitor Amyloid-β production inhibitor gammaSecretase Modulators,gamma Secretase Modulators (E)-(4R,9AS)-7-[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)benzylidene]-4-(3,4,5-trifluorophenyl)h (E)-(4R,9aS)-7-[3-Methoxy-4-(4-methyl-1H-imidazol-1-yl)benzylidene]-4-(3,4,5-trifluorophenyl)hexahydropyrido[2,1-c][1,4]oxazin-6-one hexahydro-7-[[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]methylene]-4-(3,4,5-trifluorophenyl)-(4R,7E,9aS)-Pyrido[2,1-c][1,4]oxazin-6(1H)-one Pyrido[2,1-c][1,4]oxazin-6(1H)-one, hexahydro-7-[[3-Methoxy-4-(4-Methyl-1H-iMidazol-1-yl)phenyl]Methylene]-4-(3,4,5-trifluorophenyl)-, (4R,7E,9aS)- | [Molecular Formula]
C26H24F3N3O3 | [MDL Number]
MFCD13184813 | [MOL File]
937812-80-1.mol | [Molecular Weight]
483.48 |
Chemical Properties | Back Directory | [Boiling point ]
682.5±55.0 °C(Predicted) | [density ]
1.37 | [storage temp. ]
Store at -20°C | [solubility ]
Soluble in DMSO | [form ]
Powder | [pka]
5.76±0.61(Predicted) | [color ]
White to off-white |
Hazard Information | Back Directory | [Uses]
A potent (Ki = 0.5 nM), selective, rapid acting, competitive and reversible fXa inhibitor that effectively inhibits both free and prothrombinase-bound fXa. Clinical studies show that it is efficacious, safe and well tolerated in humans and therefore has considerable potential for the treatment of acute coronary syndrome. | [storage]
Store at -20°C |
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Company Name: |
Musechem
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+1-800-259-7612 |
Website: |
www.musechem.com |
Company Name: |
BOC Sciences
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16314854226 |
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www.bocsci.com |
Company Name: |
Creative Enzymes
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Tel: |
1-516-855-7709 |
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www.creative-enzymes.com |
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