Identification | Back Directory | [Name]
Olcegepant (hydrochloride) | [CAS]
586368-06-1 | [Synonyms]
BIBN-4096 hydrochloride BIBN4096BS hydrochloride BIBN-4096BS hydrochloride BIBN 4096BS hydrochloride Olcegepant (hydrochloride) BIBN-4096 HYDROCHLORIDE; BIBN-4096BS HYDROCHLORIDE; BIBN4096BS HYDROCHLORIDE; BIBN 4096BS HYDROCHLORIDE | [Molecular Formula]
C38H48Br2ClN9O5 | [MOL File]
586368-06-1.mol | [Molecular Weight]
906.12 |
Hazard Information | Back Directory | [Biological Activity]
Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 14.4 pM for human CGRP. | [in vivo]
Olcegepant (BIBN4096BS) in doses between 1 and 30 μg/kg (i.v.) inhibits the effects of CGRP, released by stimulation of the trigeminal ganglion, on facial blood flow in marmoset monkeys. Pre-treatment with Olcegepant (900 μg/kg) inhibits the capsaicin-induced expression of Fos throughout the spinal trigeminal nucleus by 57%. | [target]
IC50: 0.03 nM (CGRP1) Ki: 14.4 pM (hCGRP) | [storage]
Store at -20°C |
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