Identification | Back Directory | [Name]
trimethyl-[4-(2-oxopyrrolidin-1-yl)but-2-ynyl]azanium:iodide | [CAS]
3854-04-4 | [Synonyms]
CPD3509 Oxotremorine M (iodide) trimethyl-[4-(2-oxopyrrolidin-1-yl)but-2-ynyl]azanium:iodide | [Molecular Formula]
C11H19IN2O | [MDL Number]
MFCD00055133 | [MOL File]
3854-04-4.mol | [Molecular Weight]
322.186 |
Chemical Properties | Back Directory | [storage temp. ]
Desiccate at -20°C | [solubility ]
DMSO : 125 mg/mL (387.97 mM; Need ultrasonic) | [form ]
Powder | [color ]
Light yellow to yellow | [Water Solubility ]
Soluble to 100 mM in water |
Hazard Information | Back Directory | [Description]
Oxotremorine M is a non-selective muscarinic (M) acetylcholine receptor agonist that induces phosphoinositide hydrolysis in mouse ileum isolated from wild-type, M2, M3, and M2/M3 knockout mice (EC50s = 0.36, 0.52, 1.62, and 1.48 μM, respectively). It also increases M4-induced inhibition of calcium currents in NG108-15 mouse neuroblastoma X rat glioma hybrid cells (EC50 = 0.14 μM). Oxotremorine M inhibits KCNQ2/3 potassium currents in Xenopus oocytes expressing M1 receptors and KCNQ2/3 potassium channels (IC50 = 1.1 μM). It also directly inhibits KCNQ2/3 potassium channels, decreasing KCNQ2/3 potassium currents in Xenopus oocytes lacking muscarinic receptors in a dose-dependent manner. | [Uses]
Oxotremorine M is a muscarinic receptor agonist. | [storage]
Desiccate at -20°C |
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BOC Sciences
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InvivoChem
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MedChemExpress
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