Identification | Back Directory | [Name]
DH 97 | [CAS]
343263-95-6 | [Synonyms]
DH 97 N-PENTANOYL-2-BENZYLTRYPTAMINE N-[2-(2-benzyl-1H-indol-3-yl)ethyl]pentanamide 1-Pentanone,1-[3-(2-aminoethyl)-2-(phenylmethyl)-1H-indol-1-yl]- | [Molecular Formula]
C22H26N2O | [MDL Number]
MFCD02262121 | [MOL File]
343263-95-6.mol | [Molecular Weight]
334.45 |
Hazard Information | Back Directory | [Description]
DH 97 is an antagonist of melatonin receptor 2 (MT2; Kis = 252 and 1,100 for human MT2 and MT1 receptors, respectively). | [Definition]
ChEBI: N-[2-[2-(phenylmethyl)-1H-indol-3-yl]ethyl]pentanamide is a member of indoles. | [Biological Activity]
A relatively potent MT 2 melatonin receptor antagonist (pK i value = 8.03), displaying 89- and 229-fold selectivity over MT 1 and GPR50 (melatonin-related orphan receptor) respectively. |
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Company Name: |
MOLEKULA Ltd.
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Tel: |
+44 (0) 1747 831066 |
Website: |
www.molekula.co.uk |
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