| Identification | Back Directory | [Name]
5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE | [CAS]
144625-67-2 | [Synonyms]
GR 125487
GR 125487 SULFAMATE
GR 125487 SULFAMATE SALT
(1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)-methyl 5-fluoro-2-methoxy-1H-indole-3-carboxyla
(1-(2-(Methylsulfonamido)ethyl)piperidin-4-yl)-methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate
5-Fluoro-2-methoxy-[1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]-1H-indole-3-methylcarboxylatesulfamate
5-fluoro-2-Methoxy-1H-Indole-3-carboxylic acid-[1-[2-[(Methylsulfonyl)aMino]ethyl]-4-piperidinyl]Methyl ester
5-FLUORO-2-METHOXY-[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]-1H-INDOLE-3-METHYLCARBOXYLATE SULFAMATE
1H-Indole-3-carboxylic acid, 5-fluoro-2-methoxy-, [1-[2-[(methylsulfonyl)amino]ethyl]-4-piperidinyl]methyl ester
[1-[2-[(METHYLSULFONYL)AMINO]ETHYL]-4-PIPERIDINYL]METHYL 5-FLUORO-2-METHOXY-1H-INDOLE-3-CARBOXYLATE SULFAMATE SALT | [Molecular Formula]
C19H26FN3O5S | [MDL Number]
MFCD00912900 | [MOL File]
144625-67-2.mol | [Molecular Weight]
427.49 |
| Chemical Properties | Back Directory | [Melting point ]
118-120℃ | [Boiling point ]
613.4±65.0 °C(Predicted) | [density ]
1.313±0.06 g/cm3(Predicted) | [storage temp. ]
Sealed in dry,2-8°C | [solubility ]
H2O: ~14 mg/mL at 60 °C, soluble | [form ]
solid | [pka]
11.22±0.40(Predicted) | [color ]
off-white |
| Hazard Information | Back Directory | [Uses]
GR 125487 Sulfamate is potent, selective 5-HT4 antagonist; active in vivo. | [Biological Activity]
Potent and selective 5-HT 4 receptor antagonist (K i = 0.19 nM for porcine 5-HT 4 ). Centrally active following systemic administration in vivo . |
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