| Identification | Back Directory | [Name]
Antihistamine-1 | [CAS]
1186430-60-3 | [Synonyms]
Antihistamine-1
1H-Benzimidazole, 1-[(4-fluorophenyl)methyl]-2-[4-(4-methyl-1H-pyrazol-1-yl)-1-piperidinyl]- | [Molecular Formula]
C23H24FN5 | [MDL Number]
MFCD30533323 | [MOL File]
1186430-60-3.mol | [Molecular Weight]
389.47 |
| Chemical Properties | Back Directory | [Boiling point ]
596.0±60.0 °C(Predicted) | [density ]
1.28±0.1 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [solubility ]
Soluble in DMSO | [form ]
Solid | [pka]
7.66±0.10(Predicted) | [color ]
Off-white to light yellow |
| Hazard Information | Back Directory | [Uses]
1-[(4-Fluorophenyl)methyl]-2-[4-(4-methyl-1H-pyrazol-1-yl)-1-piperidinyl]-1H-benzimidazole, is a 2-aminobenzimidazole H1-antihistamines used for the treatment of insomnia. It is also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM. |
|
| Company Name: |
MedChemExpress
|
| Tel: |
021-58955995 |
| Website: |
www.medchemexpress.com |
|