Identification | Back Directory | [Name]
3-Pyridinesulfonamide, 5-[8-(1H-pyrazol-4-yl)-1,5-naphthyridin-2-yl]- | [CAS]
1092565-44-0 | [Synonyms]
MMV024101 MMV-024101 MMV 024101 TCMDC134293 TCMDC-134293 TCMDC 134293 3-Pyridinesulfonamide, 5-[8-(1H-pyrazol-4-yl)-1,5-naphthyridin-2-yl]- | [Molecular Formula]
C16H12N6O2S | [MOL File]
1092565-44-0.mol | [Molecular Weight]
352.37 |
Hazard Information | Back Directory | [Description]
MMV024101 is a PI4K inhibitor. MMV024101 showed submicromolar potency against P. falciparum NF54 (IC50 =543 nM), low aqueous solubility (<5 μM), and rapid clearance by mouse liver microsomes with only 2% of parent compound remaining after 30 min of incubation. |
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